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Effect of Low-Frequency, Low-Energy Pulsed Electromagnetic Fields in Neuronal and Microglial Cells Injured with Amyloid-Beta
Merighi, Stefania; Nigro, Manuela; Travagli, Alessia; Fernandez, Mercedes; Vincenzi, Fabrizio; Varani, Katia; Pasquini, Silvia; Borea, Pier Andrea; Salati, Simona; Cadossi, Ruggero; Gessi, Stefania     dettagli >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 25, No. 1, pp: 1-21, Anno: 2024

Binding and unbinding of potent melatonin receptor ligands: Mechanistic simulations and experimental evidence
Bedini, Annalida; Elisi, Gian Marco; Fanini, Fabiola; Retini, Michele; Scalvini, Laura; Pasquini, Silvia; Contri, Chiara; Varani, Katia; Spadoni, Gilberto; Mor, Marco; Vincenzi, Fabrizio; Rivara, Silvia     dettagli >>
JOURNAL OF PINEAL RESEARCH
Vol. 76, No. 2, pp: 1-15, Anno: 2024

Spirotetrahydroisoquinoline-Based Histone Deacetylase Inhibitors as New Antifibrotic Agents: Biological Evaluation in Human Fibroblasts from Bronchoalveolar Lavages of Idiopathic Pulmonary Fibrosis Patients
Fontana, A.; Bergantini, L.; Carullo, G.; Scalvini, L.; D'Alessandro, M.; Papulino, C.; Cameli, P.; Gangi, S.; Vincenzi, F.; Varani, K.; Contri, C.; Pasquini, S.; Pistocchi, A.; Pezzotta, A.; Carbone, S.; Saponara, S.; Gemma, S.; Altucci, L.; Benedetti, R.; Lodola, A.; Mor, M.; Bargagli, E.; Butini, S.; Campiani, G.     dettagli >>
ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE
Vol. -, No. 1, pp: 1-14, Anno: 2024

Targeting Relevant HDACs to Support the Survival of Cone Photoreceptors in Inherited Retinal Diseases: Identification of a Potent Pharmacological Tool with In Vitro and In Vivo Efficacy
Carullo, G.; Orsini, N.; Piano, I.; Pozzetti, L.; Papa, A.; Fontana, A.; Napoli, D.; Corsi, F.; Marco, B. D.; Galante, A.; Marotta, L.; Panzeca, G.; O'Brien, J.; Sanchez, A. G.; Doherty, H.; Mahon, N.; Clarke, L.; Contri, C.; Pasquini, S.; Gorelli, B.; Saponara, S.; Valoti, M.; Vincenzi, F.; Varani, K.; Ramunno, A.; Brogi, S.; Butini, S.; Gemma, S.; Kennedy, B. N.; Gargini, C.; Strettoi, E.; Campiani, G.     dettagli >>
JOURNAL OF MEDICINAL CHEMISTRY
Vol. 67, No. 17, pp: 14946-14973, Anno: 2024

Synthesis and Biological Evaluation of Novel 2-Aroyl Benzofuran-Based Hydroxamic Acids as Antimicrotubule Agents
Mariotto, Elena; Canton, Martina; Marchioro, Chiara; Brancale, Andrea; Hamel, Ernest; Varani, Katia; Vincenzi, Fabrizio; De Ventura, Tiziano; Padroni, Chiara; Viola, Giampietro; Romagnoli, Romeo     dettagli >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 25, No. 14, pp: 7519-7519, Anno: 2024

Development of Epigenetic Modifiers with Therapeutic Potential in FMS-Related Tyrosine Kinase 3/Internal Tandem Duplication (FLT3/ITD) Acute Myeloid Leukemia and Other Blood Malignancies
Carullo, G.; Rossi, S.; Giudice, V.; Pezzotta, A.; Chianese, U.; Scala, P.; Carbone, S.; Fontana, A.; Panzeca, G.; Pasquini, S.; Contri, C.; Gemma, S.; Ramunno, A.; Saponara, S.; Galvani, F.; Lodola, A.; Mor, M.; Benedetti, R.; Selleri, C.; Varani, K.; Butini, S.; Altucci, L.; Vincenzi, F.; Pistocchi, A.; Campiani, G.     dettagli >>
ACS PHARMACOLOGY & TRANSLATIONAL SCIENCE
Vol. 7, No. 7, pp: 2125-2142, Anno: 2024

A novel potent class I HDAC inhibitor reverses the STAT4/p66Shc apoptotic defect in B cells from chronic lymphocytic leukemia patients
Rossi, S.; Tatangelo, V.; Dichiara, M.; Butini, S.; Gemma, S.; Brogi, S.; Pasquini, S.; Cappello, M.; Vincenzi, F.; Varani, K.; Lopresti, L.; Malchiodi, M.; Carrara, C.; Gozzetti, A.; Bocchia, M.; Marotta, G.; Patrussi, L.; Carullo, G.; Baldari, C. T.; Campiani, G.     dettagli >>
BIOMEDICINE & PHARMACOTHERAPY
Vol. 174, No. 1, pp: 1-13, Anno: 2024

Caffeine for Prevention of Alzheimer's Disease: Is the A2A Adenosine Receptor Its Target?
Merighi, Stefania; Travagli, Alessia; Nigro, Manuela; Pasquini, Silvia; Cappello, Martina; Contri, Chiara; Varani, Katia; Vincenzi, Fabrizio; Borea, Pier Andrea; Gessi, Stefania     dettagli >>
BIOMOLECULES
Vol. 13, No. 6, pp: 967-1-967-15, Anno: 2023

2-Amino-5-arylethynyl-thiophen-3-yl-(phenyl)methanones as A1 Adenosine Receptor Positive Allosteric Modulators
Oliva, Paola; Suresh, R Rama; Pasquini, Silvia; Salmaso, Veronica; Will, Edward J; Tosh, Dilip K; Gao, Zhan-Guo; Liu, Naili; Gavrilova, Oksana; Vincenzi, Fabrizio; Varani, Katia; Jacobson, Kenneth A     dettagli >>
ACS MEDICINAL CHEMISTRY LETTERS
Vol. 14, No. 12, pp: 1640-1646, Anno: 2023

Combined targeting of fatty acid amide hydrolase and melatonin receptors promotes neuroprotection and stimulates inflammation resolution in rats
Cammarota, Mariarosaria; Ferlenghi, Francesca; Vacondio, Federica; Vincenzi, Fabrizio; Varani, Katia; Bedini, Annalida; Rivara, Silvia; Mor, Marco; Boscia, Francesca     dettagli >>
BRITISH JOURNAL OF PHARMACOLOGY
Vol. 180, No. 10, pp: 1316-1338, Anno: 2023

Pharmacology of Adenosine Receptors: Recent Advancements
Vincenzi, Fabrizio; Pasquini, Silvia; Contri, Chiara; Cappello, Martina; Nigro, Manuela; Travagli, Alessia; Merighi, Stefania; Gessi, Stefania; Borea, Pier Andrea; Varani, Katia     dettagli >>
BIOMOLECULES
Vol. 13, No. 9, pp: 1387-1-1387-33, Anno: 2023

Are Two Riboses Better Than One? The Case of the Recognition and Activation of Adenosine Receptors
Gianferrara, Teresa; Pavan, Matteo; Bassani, Davide; Vincenzi, Fabrizio; Pasquini, Silvia; Bolcato, Giovanni; Varani, Katia; Spalluto, Giampiero; Federico, Stephanie; Moro, Stefano     dettagli >>
CHEMMEDCHEM
Vol. 18, No. 14, pp: e202300109-1-e202300109-14, Anno: 2023

MAM-2201 acute administration impairs motor, sensorimotor, prepulse inhibition, and memory functions in mice: a comparison with its analogue AM-2201
Corli, Giorgia; Tirri, Micaela; Bilel, Sabrine; Arfe, Raffaella; Coccini, Teresa; Roda, Elisa; Marchetti, Beatrice; Vincenzi, Fabrizio; Zauli, Giorgio; Borea, Pier Andrea; Locatelli, Carlo Alessandro; Varani, Katia; Marti, Matteo     dettagli >>
PSYCHOPHARMACOLOGY
Vol. 240, No. 7, pp: 1435-1452, Anno: 2023

Development of potent and selective FAAH inhibitors with improved drug-like properties as potential tools to treat neuroinflammatory conditions
Papa, Alessandro; Pasquini, Silvia; Galvani, Francesca; Cammarota, Mariarosaria; Contri, Chiara; Carullo, Gabriele; Gemma, Sandra; Ramunno, Anna; Lamponi, Stefania; Gorelli, Beatrice; Saponara, Simona; Varani, Katia; Mor, Marco; Campiani, Giuseppe; Boscia, Francesca; Vincenzi, Fabrizio; Lodola, Alessio; Butini, Stefania     dettagli >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 246, No. 1, pp: 114952-1-114952-22, Anno: 2023

Pioneering first-in-class FAAH-HDAC inhibitors as potential multitarget neuroprotective agents
Papa, Alessandro; Cursaro, Ilaria; Pozzetti, Luca; Contri, Chiara; Cappello, Martina; Pasquini, Silvia; Carullo, Gabriele; Ramunno, Anna; Gemma, Sandra; Varani, Katia; Butini, Stefania; Campiani, Giuseppe; Vincenzi, Fabrizio     dettagli >>
ARCHIV DER PHARMAZIE
Vol. 356, No. 12, pp: 2300410-1-2300410-22, Anno: 2023

Strategies for Drug Delivery into the Brain: A Review on Adenosine Receptors Modulation for Central Nervous System Diseases Therapy
Fernandez, M; Nigro, M; Travagli, A; Pasquini, S; Vincenzi, F; Varani, K; Borea, Pa; Merighi, S; Gessi, S     dettagli >>
PHARMACEUTICS
Vol. 15, No. 10, pp: 2441-1-2441-19, Anno: 2023

Pathophysiological Role and Medicinal Chemistry of A2A Adenosine Receptor Antagonists in Alzheimer's Disease
Merighi, Stefania; Borea, Pier Andrea; Varani, Katia; Vincenzi, Fabrizio; Travagli, Alessia; Nigro, Manuela; Pasquini, Silvia; Suresh, R Rama; Kim, Sung Won; Volkow, Nora D; Jacobson, Kenneth A; Gessi, Stefania     dettagli >>
MOLECULES
Vol. 27, No. 9, pp: 2680-1-2680-15, Anno: 2022

In Vivo Bio-Activation of JWH-175 to JWH-018: Pharmacodynamic and Pharmacokinetic Studies in Mice
Tirri, Micaela; Arfè, Raffaella; Bilel, Sabrine; Corli, Giorgia; Marchetti, Beatrice; Fantinati, Anna; Vincenzi, Fabrizio; De-Giorgio, Fabio; Camuto, Cristian; Mazzarino, Monica; Barbieri, Mario; Gaudio, Rosa Maria; Varani, Katia; Borea, Pier Andrea; Botrè, Francesco; Marti, Matteo     dettagli >>
INTERNATIONAL JOURNAL OF MOLECULAR SCIENCES
Vol. 23, No. 14, pp: 8030-1-8030-29, Anno: 2022

Pulsed Electromagnetic Fields: A Novel Attractive Therapeutic Opportunity for Neuroprotection After Acute Cerebral Ischemia
Capone, F.; Salati, S.; Vincenzi, F.; Liberti, M.; Aicardi, G.; Apollonio, F.; Varani, K.; Cadossi, R.; Di Lazzaro, V.     dettagli >>
NEUROMODULATION
Vol. 25, No. 8, pp: 1240-1247, Anno: 2022

2-Arylmelatonin analogues: Probing the 2-phenyl binding pocket of melatonin MT1 and MT2 receptors
Mari, Michele; Elisi, Gian Marco; Bedini, Annalida; Lucarini, Simone; Retini, Michele; Lucini, Valeria; Scaglione, Francesco; Vincenzi, Fabrizio; Varani, Katia; Castelli, Riccardo; Mor, Marco; Rivara, Silvia; Spadoni, Gilberto     dettagli >>
EUROPEAN JOURNAL OF MEDICINAL CHEMISTRY
Vol. 243, No. 1, pp: 1-15, Anno: 2022

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